PDB Information

PDB5FPG
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI BL21(DE3)
Gene SourceHOMO SAPIENS
Primary Citation
Design, Synthesis and Evaluation of Novel Dual- Binding Inhibitors of the Tankyrases and Wnt Signalling.
Nathubhai, A., Haikarainen, T., Hayward, P.C., Munoz-Descalzo, S., Tosh, D., Lloyd, M.D., Lehtio, L., Threadgill, M.D.
To be Published
HeaderTransferase
Released2015-11-30
Resolution2.750
CATH Insert Date08 Jan, 2017

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 09 Jan, 2017 Chopped
B 09 Jan, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5fpgA00 18 Jan, 2017 3.90.228.10 Assigned
5fpgB00 18 Jan, 2017 3.90.228.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2