PDB Information

PDB5FP3
MethodX-RAY DIFFRACTION
Host OrganismSPODOPTERA FRUGIPERDA
Gene SourceHOMO SAPIENS
Primary Citation
Cell Penetrant Inhibitors of the Kdm4 and Kdm5 Families of Histone Lysine Demethylases. 1. 3-Amino-4-Pyridine Carboxylate Derivatives.
Westaway, S.M., Preston, A.G.S., Barker, M.D., Brown, F., Brown, J.A., Campbell, M., Chung, C., Diallo, H., Douault, C., Drewes, G., Eagle, R., Gordon, L., Haslam, C., Hayhow, T.G., Humphreys, P.G., Joberty, G., Katso, R., Kruidenier, L., Leveridge, M., Liddle, J., Mosley, J., Muelbaier, M., Randle, R., Rioja, I., Rueger, A., Seal, G.A., Sheppard, R.J., Singh, O., Taylor, J., Thomas, P., Thomson, D., Wilson, D.M., Lee, K., Prinjha, R.K.
J.Med.Chem.
HeaderOxidoreductase
Released2015-11-27
Resolution2.050
CATH Insert Date10 Apr, 2016

PDB Images (9)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Chopped
B 11 Apr, 2016 Chopped

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
5fp3A01 11 May, 2016 2.60.120.650 Assigned
5fp3A02 11 May, 2016 1.20.58.1370 Assigned
5fp3A03 11 May, 2016 2.10.110.20 Assigned
5fp3B01 11 May, 2016 2.60.120.650 Assigned
5fp3B02 11 May, 2016 1.20.58.1370 Assigned
5fp3B03 11 May, 2016 2.10.110.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O15054 KDM6B_HUMAN Homo sapiens Lysine-specific demethylase 6B
O15054 KDM6B_HUMAN Homo sapiens Lysine-specific demethylase 6B