PDB Information

PDB5FI7
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design and evaluation of novel glutaminase inhibitors.
McDermott, L.A., Iyer, P., Vernetti, L., Rimer, S., Sun, J., Boby, M., Yang, T., Fioravanti, M., O'Neill, J., Wang, L., Drakes, D., Katt, W., Huang, Q., Cerione, R.
Bioorg.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2015-12-22
Resolution2.500
CATH Insert Date29 May, 2016

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 30 May, 2016 Chopped
B 30 May, 2016 Chopped
C 30 May, 2016 Chopped
D 30 May, 2016 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5fi7A01 16 Jul, 2016 1.10.238.210 Assigned
5fi7A02 16 Jul, 2016 3.40.710.10 Assigned
5fi7B01 16 Jul, 2016 1.10.238.210 Assigned
5fi7B02 16 Jul, 2016 3.40.710.10 Assigned
5fi7C01 16 Jul, 2016 1.10.238.210 Assigned
5fi7C02 16 Jul, 2016 3.40.710.10 Assigned
5fi7D01 16 Jul, 2016 1.10.238.210 Assigned
5fi7D02 16 Jul, 2016 3.40.710.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial