PDB Information

PDB5FI2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design and evaluation of novel glutaminase inhibitors.
McDermott, L.A., Iyer, P., Vernetti, L., Rimer, S., Sun, J., Boby, M., Yang, T., Fioravanti, M., O'Neill, J., Wang, L., Drakes, D., Katt, W., Huang, Q., Cerione, R.
Bioorg.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2015-12-22
Resolution2.500
CATH Insert Date29 May, 2016

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 30 May, 2016 Chopped
B 30 May, 2016 Chopped
C 30 May, 2016 Chopped
D 30 May, 2016 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5fi2A01 15 Jul, 2016 1.10.238.210 Assigned
5fi2A02 15 Jul, 2016 3.40.710.10 Assigned
5fi2B01 16 Jul, 2016 1.10.238.210 Assigned
5fi2B02 16 Jul, 2016 3.40.710.10 Assigned
5fi2C01 16 Jul, 2016 1.10.238.210 Assigned
5fi2C02 16 Jul, 2016 3.40.710.10 Assigned
5fi2D01 16 Jul, 2016 1.10.238.210 Assigned
5fi2D02 16 Jul, 2016 3.40.710.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial