PDB 5f9e
PDB Information
| PDB | 5F9E |
| Method | X-RAY DIFFRACTION |
| Host Organism | unidentified baculovirus |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery and optimization of 1,7-disubstituted-2,2-dimethyl-2,3-dihydroquinazolin-4(1H)-ones as potent and selective PKC theta inhibitors.
Bioorg.Med.Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2015-12-09 |
| Resolution | 2.000 |
| CATH Insert Date | 29 May, 2016 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 30 May, 2016 | Chopped |
| B | 30 May, 2016 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5f9eA01 | 15 Jul, 2016 | 3.30.200.20 | Assigned |
| 5f9eA02 | 15 Jul, 2016 | 1.10.510.10 | Assigned |
| 5f9eB01 | 15 Jul, 2016 | 3.30.200.20 | Assigned |
| 5f9eB02 | 15 Jul, 2016 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q04759 | KPCT_HUMAN | Homo sapiens | Protein kinase C theta type |
| Q04759 | KPCT_HUMAN | Homo sapiens | Protein kinase C theta type |
