PDB 5f95
PDB Information
| PDB | 5F95 |
| Method | X-RAY DIFFRACTION |
| Host Organism | unidentified baculovirus |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of Isonicotinamides as Highly Selective, Brain Penetrable, and Orally Active Glycogen Synthase Kinase-3 Inhibitors.
J.Med.Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2015-12-09 |
| Resolution | 2.530 |
| CATH Insert Date | 10 Apr, 2016 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 11 Apr, 2016 | Chopped |
| B | 11 Apr, 2016 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5f95A01 | 10 May, 2016 | 3.30.200.20 | Assigned |
| 5f95A02 | 10 May, 2016 | 1.10.510.10 | Assigned |
| 5f95B01 | 10 May, 2016 | 3.30.200.20 | Assigned |
| 5f95B02 | 10 May, 2016 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P49841 | GSK3B_HUMAN | Homo sapiens | Glycogen synthase kinase-3 beta |
| P49841 | GSK3B_HUMAN | Homo sapiens | Glycogen synthase kinase-3 beta |
