PDB Information

PDB5F92
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMycobacterium tuberculosis (strain CDC 1551 / Oshkosh)
Primary Citation
Selective small molecule inhibitor of the Mycobacterium tuberculosis fumarate hydratase reveals an allosteric regulatory site.
Kasbekar, M., Fischer, G., Mott, B.T., Yasgar, A., Hyvonen, M., Boshoff, H.I., Abell, C., Barry, C.E., Thomas, C.J.
Proc.Natl.Acad.Sci.USA
HeaderLyase
Released2015-12-09
Resolution1.860
CATH Insert Date10 Jul, 2016

PDB Images (17)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 11 Jul, 2016 Chopped
B 11 Jul, 2016 Chopped
C 11 Jul, 2016 Chopped
D 11 Jul, 2016 Chopped

CATH Domains (12)

Domain ID Date inserted into CATH Superfamily CATH Status
5f92A01 15 Jul, 2016 1.10.275.10 Assigned
5f92A02 15 Jul, 2016 1.20.200.10 Assigned
5f92A03 15 Jul, 2016 1.10.40.30 Assigned
5f92B01 15 Jul, 2016 1.10.275.10 Assigned
5f92B02 15 Jul, 2016 1.20.200.10 Assigned
5f92B03 15 Jul, 2016 1.10.40.30 Assigned
5f92C01 15 Jul, 2016 1.10.275.10 Assigned
5f92C02 15 Jul, 2016 1.20.200.10 Assigned
5f92C03 15 Jul, 2016 1.10.40.30 Assigned
5f92D01 15 Jul, 2016 1.10.275.10 Assigned
5f92D02 15 Jul, 2016 1.20.200.10 Assigned
5f92D03 15 Jul, 2016 1.10.40.30 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P9WN92 FUMC_MYCTO Mycobacterium tuberculosis CDC1551 Fumarate hydratase class II
P9WN92 FUMC_MYCTO Mycobacterium tuberculosis CDC1551 Fumarate hydratase class II
P9WN92 FUMC_MYCTO Mycobacterium tuberculosis CDC1551 Fumarate hydratase class II
P9WN92 FUMC_MYCTO Mycobacterium tuberculosis CDC1551 Fumarate hydratase class II