PDB Information

PDB5F61
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Potent Dual BET Bromodomain-Kinase Inhibitors as Value-Added Multitargeted Chemical Probes and Cancer Therapeutics.
Ember, S.W., Lambert, Q.T., Berndt, N., Gunawan, S., Ayaz, M., Tauro, M., Zhu, J.Y., Cranfill, P.J., Greninger, P., Lynch, C.C., Benes, C.H., Lawrence, H.R., Reuther, G.W., Lawrence, N.J., Schonbrunn, E.
Mol. Cancer Ther.
HeaderTranscription/Transcription Inhibitor
Released2015-12-04
Resolution1.450
CATH Insert Date07 May, 2017

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5f61A01 12 May, 2017 1.20.920.10 Assigned
5f61B01 12 May, 2017 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4