PDB Information

PDB5F25
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor.
Martin, L.J., Koegl, M., Bader, G., Cockcroft, X.L., Fedorov, O., Fiegen, D., Gerstberger, T., Hofmann, M.H., Hohmann, A.F., Kessler, D., Knapp, S., Knesl, P., Kornigg, S., Muller, S., Nar, H., Rogers, C., Rumpel, K., Schaaf, O., Steurer, S., Tallant, C., Vakoc, C.R., Zeeb, M., Zoephel, A., Pearson, M., Boehmelt, G., McConnell, D.
J.Med.Chem.
HeaderTranscription
Released2015-12-01
Resolution1.680
CATH Insert Date10 Apr, 2016

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Chopped
B 11 Apr, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5f25A00 09 May, 2016 1.20.920.10 Assigned
5f25B00 09 May, 2016 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9H8M2 BRD9_HUMAN Homo sapiens Bromodomain-containing protein 9
Q9H8M2 BRD9_HUMAN Homo sapiens Bromodomain-containing protein 9