PDB Information

PDB5EZG
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMycobacterium tuberculosis
Primary Citation
A fragment merging approach towards the development of small molecule inhibitors of Mycobacterium tuberculosis EthR for use as ethionamide boosters.
Nikiforov, P.O., Surade, S., Blaszczyk, M., Delorme, V., Brodin, P., Baulard, A.R., Blundell, T.L., Abell, C.
Org.Biomol.Chem.
HeaderTranscription
Released2015-11-26
Resolution1.840
CATH Insert Date10 Apr, 2016

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5ezgA01 09 May, 2016 1.10.10.60 Assigned
5ezgA02 09 May, 2016 1.10.357.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P9WMC0 ETHR_MYCTO Mycobacterium tuberculosis CDC1551 HTH-type transcriptional regulator EthR