PDB 5eym
PDB Information
| PDB | 5EYM |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Pharmacological Profile of BI 847325, an Orally Bioavailable, ATP-Competitive Inhibitor of MEK and Aurora Kinases.
Mol.Cancer Ther.
|
| Header | Transferase |
| Released | 2015-11-25 |
| Resolution | 2.700 |
| CATH Insert Date | 04 Sep, 2016 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 05 Sep, 2016 | Chopped |
| B | 05 Sep, 2016 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5eymA01 | 09 Sep, 2016 | 3.30.200.20 | Assigned |
| 5eymA02 | 09 Sep, 2016 | 1.10.510.10 | Assigned |
| 5eymB01 | 08 Sep, 2016 | 3.30.200.20 | Assigned |
| 5eymB02 | 08 Sep, 2016 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q02750 | MP2K1_HUMAN | Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 1 |
| Q02750 | MP2K1_HUMAN | Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 1 |
