PDB Information

PDB5ETY
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
The Discovery and Characterization of K-756, a Novel Wnt/ beta-Catenin Pathway Inhibitor Targeting Tankyrase
Okada-Iwasaki, R., Takahashi, Y., Watanabe, Y., Ishida, H., Saito, J., Nakai, R., Asai, A.
Mol.Cancer Ther.
HeaderTransferase
Released2015-11-18
Resolution2.900
CATH Insert Date10 Jul, 2016

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 11 Jul, 2016 Chopped
B 11 Jul, 2016 Chopped
C 11 Jul, 2016 Chopped
D 11 Jul, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5etyA00 15 Jul, 2016 3.90.228.10 Assigned
5etyB00 15 Jul, 2016 3.90.228.10 Assigned
5etyC00 15 Jul, 2016 3.90.228.10 Assigned
5etyD00 15 Jul, 2016 3.90.228.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
O95271 TNKS1_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-1
O95271 TNKS1_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-1
O95271 TNKS1_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-1
O95271 TNKS1_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-1