PDB Information

PDB5EGU
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Exploring Selective Inhibition of the First Bromodomain of the Human Bromodomain and Extra-terminal Domain (BET) Proteins.
Raux, B., Voitovich, Y., Derviaux, C., Lugari, A., Rebuffet, E., Milhas, S., Priet, S., Roux, T., Trinquet, E., Guillemot, J.C., Knapp, S., Brunel, J.M., Fedorov, A.Y., Collette, Y., Roche, P., Betzi, S., Combes, S., Morelli, X.
J.Med.Chem.
HeaderTranscription
Released2015-10-27
Resolution2.210
CATH Insert Date10 Apr, 2016

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Chopped
B 11 Apr, 2016 Chopped
C 11 Apr, 2016 Chopped
D 11 Apr, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5eguA01 08 May, 2016 1.20.920.10 Assigned
5eguB01 08 May, 2016 1.20.920.10 Assigned
5eguC01 08 May, 2016 1.20.920.10 Assigned
5eguD01 08 May, 2016 1.20.920.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4