PDB 5egu
PDB Information
PDB | 5EGU |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli BL21(DE3) |
Gene Source | Homo sapiens |
Primary Citation | Exploring Selective Inhibition of the First Bromodomain of the Human Bromodomain and Extra-terminal Domain (BET) Proteins.
J.Med.Chem.
|
Header | Transcription |
Released | 2015-10-27 |
Resolution | 2.210 |
CATH Insert Date | 10 Apr, 2016 |
PDB Images (9)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 11 Apr, 2016 | Chopped |
B | 11 Apr, 2016 | Chopped |
C | 11 Apr, 2016 | Chopped |
D | 11 Apr, 2016 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5eguA01 | 08 May, 2016 | 1.20.920.10 | Assigned |
5eguB01 | 08 May, 2016 | 1.20.920.10 | Assigned |
5eguC01 | 08 May, 2016 | 1.20.920.10 | Assigned |
5eguD01 | 08 May, 2016 | 1.20.920.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |