PDB 5edp
PDB Information
| PDB | 5EDP |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | 4-Aminoindazolyl-dihydrofuro[3,4-d]pyrimidines as non-covalent inhibitors of mutant epidermal growth factor receptor tyrosine kinase.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2015-10-21 |
| Resolution | 2.900 |
| CATH Insert Date | 20 Dec, 2015 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 21 Dec, 2015 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5edpA01 | 05 Jan, 2016 | 3.30.200.20 | Assigned |
| 5edpA02 | 05 Jan, 2016 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P00533 | EGFR_HUMAN | Homo sapiens | Epidermal growth factor receptor |
