PDB Information

PDB5E8R
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
A Potent, Selective, and Cell-Active Inhibitor of Human Type I Protein Arginine Methyltransferases.
Eram, M.S., Shen, Y., Szewczyk, M.M., Wu, H., Senisterra, G., Li, F., Butler, K.V., Kaniskan, H.U., Speed, B.A., Dela Sena, C., Dong, A., Zeng, H., Schapira, M., Brown, P.J., Arrowsmith, C.H., Barsyte-Lovejoy, D., Liu, J., Vedadi, M., Jin, J.
Acs Chem.Biol.
HeaderTransferase
Released2015-10-14
Resolution2.550
CATH Insert Date20 Dec, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 21 Dec, 2015 Chopped
B 21 Dec, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5e8rA01 20 Mar, 2016 3.40.50.150 Assigned
5e8rA02 20 Mar, 2016 2.70.160.11 Assigned
5e8rB01 20 Mar, 2016 3.40.50.150 Assigned
5e8rB02 20 Mar, 2016 2.70.160.11 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q96LA8 ANM6_HUMAN Homo sapiens Protein arginine N-methyltransferase 6
Q96LA8 ANM6_HUMAN Homo sapiens Protein arginine N-methyltransferase 6