PDB 5dey
PDB Information
| PDB | 5DEY |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Design of Selective PAK1 Inhibitor G-5555: Improving Properties by Employing an Unorthodox Low-pK a Polar Moiety.
Acs Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2015-08-26 |
| Resolution | 2.100 |
| CATH Insert Date | 10 Apr, 2016 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 11 Apr, 2016 | Chopped |
| B | 11 Apr, 2016 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5deyA01 | 07 May, 2016 | 3.30.200.20 | Assigned |
| 5deyA02 | 07 May, 2016 | 1.10.510.10 | Assigned |
| 5deyB01 | 07 May, 2016 | 3.30.200.20 | Assigned |
| 5deyB02 | 07 May, 2016 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q13153 | PAK1_HUMAN | Homo sapiens | Serine/threonine-protein kinase PAK 1 |
| Q13153 | PAK1_HUMAN | Homo sapiens | Serine/threonine-protein kinase PAK 1 |
