PDB Information

PDB5CR5
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery, SAR, and X-ray Binding Mode Study of BCATm Inhibitors from a Novel DNA-Encoded Library.
Deng, H., Zhou, J., Sundersingh, F.S., Summerfield, J., Somers, D., Messer, J.A., Satz, A.L., Ancellin, N., Arico-Muendel, C.C., Sargent Bedard, K.L., Beljean, A., Belyanskaya, S.L., Bingham, R., Smith, S.E., Boursier, E., Carter, P., Centrella, P.A., Clark, M.A., Chung, C.W., Davie, C.P., Delorey, J.L., Ding, Y., Franklin, G.J., Grady, L.C., Herry, K., Hobbs, C., Kollmann, C.S., Morgan, B.A., Pothier Kaushansky, L.J., Zhou, Q.
Acs Med.Chem.Lett.
HeaderTransferase
Released2015-07-22
Resolution1.610
CATH Insert Date30 Aug, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 31 Aug, 2015 Chopped
B 31 Aug, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5cr5A01 03 Sep, 2015 3.30.470.10 Assigned
5cr5A02 03 Sep, 2015 3.20.10.10 Assigned
5cr5B01 02 Sep, 2015 3.30.470.10 Assigned
5cr5B02 02 Sep, 2015 3.20.10.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O15382 BCAT2_HUMAN Homo sapiens Branched-chain-amino-acid aminotransferase, mitochondrial
O15382 BCAT2_HUMAN Homo sapiens Branched-chain-amino-acid aminotransferase, mitochondrial