PDB Information

PDB5CFW
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities.
Chekler, E.L., Pellegrino, J.A., Lanz, T.A., Denny, R.A., Flick, A.C., Coe, J., Langille, J., Basak, A., Liu, S., Stock, I.A., Sahasrabudhe, P., Bonin, P.D., Lee, K., Pletcher, M.T., Jones, L.H.
Chem.Biol.
HeaderTranscription/Inhibitor
Released2015-07-08
Resolution1.150
CATH Insert Date24 Apr, 2016

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 25 Apr, 2016 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5cfwA01 05 May, 2016 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4