PDB Information

PDB5C42
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman immunodeficiency virus type 1 group M subtype B (isolate BH10)
Primary Citation
Potent Inhibitors Active against HIV Reverse Transcriptase with K101P, a Mutation Conferring Rilpivirine Resistance.
Gray, W.T., Frey, K.M., Laskey, S.B., Mislak, A.C., Spasov, K.A., Lee, W.G., Bollini, M., Siliciano, R.F., Jorgensen, W.L., Anderson, K.S.
Acs Med.Chem.Lett.
HeaderTransferase, Hydrolase/Inhibitor
Released2015-06-17
Resolution3.500
CATH Insert Date29 Nov, 2015

PDB Images (12)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 30 Nov, 2015 Chopped
B 30 Nov, 2015 Chopped

CATH Domains (9)

Domain ID Date inserted into CATH Superfamily CATH Status
5c42A01 03 Dec, 2015 3.10.10.10 Assigned
5c42A02 03 Dec, 2015 3.30.70.270 Assigned
5c42A03 03 Dec, 2015 3.30.70.270 Assigned
5c42A04 03 Dec, 2015 3.30.70.270 Assigned
5c42A05 03 Dec, 2015 3.30.420.10 Assigned
5c42B01 03 Dec, 2015 3.10.10.10 Assigned
5c42B02 03 Dec, 2015 3.30.70.270 Assigned
5c42B03 03 Dec, 2015 3.30.70.270 Assigned
5c42B04 03 Dec, 2015 3.30.70.270 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P03366 POL_HV1B1 Human immunodeficiency virus type 1 BH10 Gag-Pol polyprotein
P03366 POL_HV1B1 Human immunodeficiency virus type 1 BH10 Gag-Pol polyprotein