PDB Information

PDB5BMS
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-Guided Design of Group I Selective p21-Activated Kinase Inhibitors.
Crawford, J.J., Lee, W., Aliagas, I., Mathieu, S., Hoeflich, K.P., Zhou, W., Wang, W., Rouge, L., Murray, L., La, H., Liu, N., Fan, P.W., Cheong, J., Heise, C.E., Ramaswamy, S., Mintzer, R., Liu, Y., Chao, Q., Rudolph, J.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2015-05-22
Resolution2.900
CATH Insert Date16 Aug, 2015

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 17 Aug, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5bmsA01 24 Aug, 2015 3.30.200.20 Assigned
5bmsA02 24 Aug, 2015 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O96013 PAK4_HUMAN Homo sapiens Serine/threonine-protein kinase PAK 4