PDB Information

PDB5BML
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Design, Synthesis, and Structure-Activity Relationships of Pyridine-Based Rho Kinase (ROCK) Inhibitors.
Green, J., Cao, J., Bandarage, U.K., Gao, H., Court, J., Marhefka, C., Jacobs, M., Taslimi, P., Newsome, D., Nakayama, T., Shah, S., Rodems, S.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2015-05-22
Resolution2.950
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5bmlA01 07 Mar, 2018 3.30.200.20 Assigned
5bmlA02 07 Mar, 2018 1.10.510.10 Assigned
5bmlB01 07 Mar, 2018 3.30.200.20 Assigned
5bmlB02 07 Mar, 2018 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q13464 ROCK1_HUMAN Homo sapiens Rho-associated protein kinase 1
Q13464 ROCK1_HUMAN Homo sapiens Rho-associated protein kinase 1