PDB 5b5p
PDB Information
| PDB | 5B5P |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21(DE3) |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of Novel, Highly Potent, and Selective Matrix Metalloproteinase (MMP)-13 Inhibitors with a 1,2,4-Triazol-3-yl Moiety as a Zinc Binding Group Using a Structure-Based Design Approach
J. Med. Chem.
|
| Header | Hydrolase/Hydrolase Inhibitor |
| Released | 2016-05-13 |
| Resolution | 1.600 |
| CATH Insert Date | 07 May, 2017 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 May, 2017 | Chopped |
| B | 08 May, 2017 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5b5pA00 | 12 May, 2017 | 3.40.390.10 | Assigned |
| 5b5pB00 | 12 May, 2017 | 3.40.390.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P45452 | MMP13_HUMAN | Homo sapiens | Collagenase 3 |
| P45452 | MMP13_HUMAN | Homo sapiens | Collagenase 3 |
