PDB Information

PDB5AYF
MethodX-RAY DIFFRACTION
Host OrganismCell-free synthesis
Gene SourceHomo sapiens
Primary Citation
Identification of Cyproheptadine as an Inhibitor of SET Domain Containing Lysine Methyltransferase 7/9 (Set7/9) That Regulates Estrogen-Dependent Transcription
Takemoto, Y., Ito, A., Niwa, H., Okamura, M., Fujiwara, T., Hirano, T., Handa, N., Umehara, T., Sonoda, T., Ogawa, K., Tariq, M., Nishino, N., Dan, S., Kagechika, H., Yamori, T., Yokoyama, S., Yoshida, M.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2015-08-20
Resolution2.010
CATH Insert Date08 May, 2016

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 09 May, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5ayfA01 12 Jul, 2016 2.20.110.10 Assigned
5ayfA02 12 Jul, 2016 2.170.270.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q8WTS6 SETD7_HUMAN Homo sapiens Histone-lysine N-methyltransferase SETD7