PDB Information

PDB5AX3
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21
Gene SourceHomo sapiens
Primary Citation
Identification of allosteric ERK2 inhibitors through in silico biased screening and competitive binding assay
Kinoshita, T., Sugiyama, H., Mori, Y., Takahashi, N., Tomonaga, A.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2015-07-14
Resolution2.980
CATH Insert Date10 Apr, 2016

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Chopped
B 11 Apr, 2016 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5ax3A01 04 May, 2016 3.30.200.20 Assigned
5ax3A02 04 May, 2016 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P28482 MK01_HUMAN Homo sapiens Mitogen-activated protein kinase 1
P40763 STAT3_HUMAN Homo sapiens Signal transducer and activator of transcription 3