PDB Information

PDB5ARG
MethodX-RAY DIFFRACTION
Host OrganismSPODOPTERA FRUGIPERDA
Gene SourceHOMO SAPIENS
Primary Citation
Discovery and Characterization of a Highly Potent and Selective Aminopyrazoline-Based in Vivo Probe (Bay-598) for the Protein Lysine Methyltransferase Smyd2.
Eggert, E., Hillig, R.C., Kohr, S., Stockigt, D., Weiske, J., Barak, N., Mowat, J., Brumby, T., Christ, C.D., Ter Laak, A., Lang, T., Fernandez-Montalvan, A.E., Badock, V., Weinmann, H., Hartung, I.V., Barsyte-Lovejoy, D., Szewczyk, M., Kennedy, S., Li, F., Vedadi, M., Brown, P.J., Santhakumar, V., Arrowsmith, C.H., Stellfeld, T., Stresemann, C.
J.Med.Chem.
HeaderTransferase
Released2015-09-24
Resolution1.990
CATH Insert Date08 May, 2016

PDB Images (5)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 09 May, 2016 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
5argA01 12 Jul, 2016 2.170.270.10 Assigned
5argA02 12 Jul, 2016 Holding pen
5argA03 12 Jul, 2016 1.25.40.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9NRG4 SMYD2_HUMAN Homo sapiens N-lysine methyltransferase SMYD2