PDB Information

PDB5AK2
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Investigation of (E)-3-[4-(2-Oxo-3-Aryl-Chromen-4-Yl)Oxyphenyl]Acrylic Acids as Oral Selective Estrogen Receptor Down-Regulators.
Degorce, S.L., Bailey, A., Callis, R., De Savi, C., Ducray, R., Lamont, G., Macfaul, P., Maudet, M., Martin, S., Morgentin, R., Norman, R.A., Peru, A., Pink, J.H., Ple, P.A., Roberts, B., Scott, J.S.
J.Med.Chem.
HeaderSignaling Protein
Released2015-02-27
Resolution2.190
CATH Insert Date28 Jun, 2015

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5ak2A00 27 Jul, 2015 1.10.565.10 Assigned
5ak2B00 27 Jul, 2015 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P03372 ESR1_HUMAN Homo sapiens Estrogen receptor
P03372 ESR1_HUMAN Homo sapiens Estrogen receptor