PDB Information

PDB5AJV
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Structure-Based Design of Potent and Selective Inhibitors of the Metabolic Kinase Pfkfb3.
Boyd, S., Brookfield, J.L., Critchlow, S.E., Cumming, I.A., Curtis, N.J., Debreczeni, J., Degorce, S.L., Donald, C., Evans, N.J., Groombridge, S., Hopcroft, P., Jones, N.P., Kettle, J.G., Lamont, S., Lewis, H.J., Macfaull, P., Mcloughlin, S.B., Rigoreau, L.J.M., Smith, J.M., St-Gallay, S., Stock, J.K., Turnbull, A.P., Wheatley, E.R., Winter, J., Wingfield, J.
J.Med.Chem.
HeaderTransferase
Released2015-02-27
Resolution3.010
CATH Insert Date28 Jun, 2015

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
B 29 Jun, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5ajvB01 27 Jul, 2015 3.40.50.300 Assigned
5ajvB02 27 Jul, 2015 3.40.50.1240 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q16875 F263_HUMAN Homo sapiens 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3