PDB 5a86
PDB Information
| PDB | 5A86 |
| Method | X-RAY DIFFRACTION |
| Host Organism | ESCHERICHIA COLI |
| Gene Source | HOMO SAPIENS |
| Primary Citation | Identification and Optimization of Benzimidazole Sulfonamides as Orally Bioavailable Sphingosine 1-Phosphate Receptor 1 Antagonists with in Vivo Activity.
J.Med.Chem.
|
| Header | Signaling Protein |
| Released | 2015-07-13 |
| Resolution | 2.250 |
| CATH Insert Date | 08 Nov, 2015 |
PDB Images (7)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 09 Nov, 2015 | Chopped |
| B | 09 Nov, 2015 | Chopped |
| C | 09 Nov, 2015 | Rejected |
| D | 09 Nov, 2015 | Rejected |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5a86A00 | 18 Nov, 2015 | 1.10.565.10 | Assigned |
| 5a86B00 | 23 Nov, 2015 | 1.10.565.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O75469 | NR1I2_HUMAN | Homo sapiens | Nuclear receptor subfamily 1 group I member 2 |
| Q15788 | NCOA1_HUMAN | Homo sapiens | Nuclear receptor coactivator 1 |
| O75469 | NR1I2_HUMAN | Homo sapiens | Nuclear receptor subfamily 1 group I member 2 |
| Q15788 | NCOA1_HUMAN | Homo sapiens | Nuclear receptor coactivator 1 |
