PDB Information

PDB5A4T
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Probing the ATP-Binding Pocket of Protein Kinase Dyrk1A with Benzothiazole Fragment Molecules
Rothweiler, U., Stensen, W., Brandsdal, B.O., Isaksson, J., Leeson, F.A., Eugh, R.A., Mjoen Svendsen, J.S.
J.Med.Chem.
HeaderTransferase
Released2015-06-15
Resolution2.150
CATH Insert Date10 Jul, 2016

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 11 Jul, 2016 Chopped
B 11 Jul, 2016 Chopped
C 11 Jul, 2016 Chopped
D 11 Jul, 2016 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5a4tA01 30 Nov, 2016 3.30.200.20 Assigned
5a4tA02 30 Nov, 2016 1.10.510.10 Assigned
5a4tB01 30 Nov, 2016 3.30.200.20 Assigned
5a4tB02 30 Nov, 2016 1.10.510.10 Assigned
5a4tC01 30 Nov, 2016 3.30.200.20 Assigned
5a4tC02 30 Nov, 2016 1.10.510.10 Assigned
5a4tD01 30 Nov, 2016 3.30.200.20 Assigned
5a4tD02 30 Nov, 2016 1.10.510.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A