PDB Information

PDB5A3U
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Potent and Selective Triazole-Based Inhibitors of the Hypoxia-Inducible Factor Prolyl-Hydroxylases with Activity in the Murine Brain.
Chan, M.C., Atasoylu, O., Hodson, E., Tumber, A., Leung, I.K.H., Chowdhury, R., Gomez-Perez, V., Demetriades, M., Rydzik, A.M., Holt-Martyn, J., Tian, Y., Bishop, T., Claridge, T.D.W., Kawamura, A., Pugh, C.W., Ratcliffe, P.J., Schofield, C.J.
Plos One
HeaderOxidoreductase
Released2015-06-03
Resolution3.300
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped
C 29 Jun, 2015 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
5a3uA00 20 Mar, 2016 2.60.120.620 Assigned
5a3uB00 27 Jul, 2015 2.60.120.620 Assigned
5a3uC00 27 Jul, 2015 2.60.120.620 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
Q9GZT9 EGLN1_HUMAN Homo sapiens Egl nine homolog 1
Q9GZT9 EGLN1_HUMAN Homo sapiens Egl nine homolog 1
Q9GZT9 EGLN1_HUMAN Homo sapiens Egl nine homolog 1