PDB 5a2s

PDB Information

PDB5A2S
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Potent, Selective, and Cns-Penetrant Tetrasubstituted Cyclopropane Class Iia Histone Deacetylase (Hdac) Inhibitors.
Luckhurst, C.A., Breccia, P., Stott, A.J., Aziz, O., Birch, H.L., Burli, R.W., Hughes, S.J., Jarvis, R.E., Lamers, M., Leonard, P.M., Matthews, K.L., Mcallister, G., Pollack, S., Saville-Stones, E., Wishart, G., Yates, D., Dominguez, C.
Acs Med.Chem.Lett.
HeaderHydrolase
Released2015-05-22
Resolution2.650
CATH Insert Date10 Apr, 2016

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Chopped
B 11 Apr, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5a2sA00 03 May, 2016 3.40.800.20 Assigned
5a2sB00 03 May, 2016 3.40.800.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P56524 HDAC4_HUMAN Homo sapiens Histone deacetylase 4
P56524 HDAC4_HUMAN Homo sapiens Histone deacetylase 4