PDB Information

PDB4ZZM
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Structure-Guided Design of Highly Selective and Potent Covalent Inhibitors of Erk1/2.
Ward, R.A., Colclough, N., Challinor, M., Debreczeni, J., Eckersley, K., Fairley, G., Feron, L., Flemington, V., Graham, M.A., Greenwood, R., Hopcroft, P., Howard, T.D., James, M., Jones, C.D., Jones, C.R., Renshaw, J., Roberts, K., Snow, L., Tonge, M., Yeung, K.
J.Med.Chem.
HeaderTransferase
Released2015-04-10
Resolution1.890
CATH Insert Date28 Jun, 2015

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4zzmA01 27 Jul, 2015 3.30.200.20 Assigned
4zzmA02 27 Jul, 2015 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P28482 MK01_HUMAN Homo sapiens Mitogen-activated protein kinase 1