PDB Information

PDB4ZY4
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-Guided Design of Group I Selective p21-Activated Kinase Inhibitors.
Crawford, J.J., Lee, W., Aliagas, I., Mathieu, S., Hoeflich, K.P., Zhou, W., Wang, W., Rouge, L., Murray, L., La, H., Liu, N., Fan, P.W., Cheong, J., Heise, C.E., Ramaswamy, S., Mintzer, R., Liu, Y., Chao, Q., Rudolph, J.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2015-05-21
Resolution2.600
CATH Insert Date16 Aug, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 17 Aug, 2015 Chopped
B 17 Aug, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4zy4A01 24 Aug, 2015 3.30.200.20 Assigned
4zy4A02 24 Aug, 2015 1.10.510.10 Assigned
4zy4B01 24 Aug, 2015 3.30.200.20 Assigned
4zy4B02 24 Aug, 2015 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q13153 PAK1_HUMAN Homo sapiens Serine/threonine-protein kinase PAK 1
Q13153 PAK1_HUMAN Homo sapiens Serine/threonine-protein kinase PAK 1