PDB Information

PDB4ZX1
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Mapping Selective Inhibition of the Cancer-Related Carbonic Anhydrase IX using Structure-Activity Relationships of Glucosyl-Based Sulfamates
Mahon, B.P., Lomelino, C.L., Moeker, J., Rankin, G.M., Driscoll, J.M., Salguero, A.L., Pinard, M.A., Vullo, D., Supuran, C.T., Poulsen, S.A., McKenna, R.
J. Med. Chem.
HeaderLyase/Lyase Inhibitor
Released2015-05-20
Resolution1.500
CATH Insert Date08 Nov, 2015

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 09 Nov, 2015 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4zx1A00 12 Nov, 2015 3.10.200.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P00918 CAH2_HUMAN Homo sapiens Carbonic anhydrase 2