PDB Information

PDB4ZTJ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman spumaretrovirus
Primary Citation
Discovery of 2-Pyridinone Aminals: A Prodrug Strategy to Advance a Second Generation of HIV-1 Integrase Strand Transfer Inhibitors.
Raheem, I.T., Walji, A.M., Klein, D., Sanders, J.M., Powell, D.A., Abeywickrema, P., Barbe, G., Bennet, A., Clas, S.D., Dubost, D., Embrey, M., Grobler, J., Hafey, M.J., Hartingh, T.J., Hazuda, D.J., Miller, M.D., Moore, K.P., Pajkovic, N., Patel, S., Rada, V., Rearden, P., Schreier, J.D., Sisko, J., Steele, T.G., Truchon, J.F., Wai, J., Xu, M., Coleman, P.J.
J.Med.Chem.
HeaderTransferase/Dna/Inhibitor
Released2015-05-14
Resolution2.670
CATH Insert Date18 Oct, 2015

PDB Images (10)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 19 Oct, 2015 Chopped
B 19 Oct, 2015 Chopped
C 19 Oct, 2015 Rejected
D 19 Oct, 2015 Rejected

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
4ztjA01 01 Nov, 2015 1.10.340.70 Assigned
4ztjA02 01 Nov, 2015 2.30.30.140 Assigned
4ztjA03 01 Nov, 2015 3.30.420.10 Assigned
4ztjA04 01 Nov, 2015 6.10.20.110 Assigned
4ztjB00 31 Oct, 2015 3.30.420.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P14350 POL_FOAMV Human spumaretrovirus Pro-Pol polyprotein
P14350 POL_FOAMV Human spumaretrovirus Pro-Pol polyprotein