PDB 4zsa
PDB Information
| PDB | 4ZSA |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Design, synthesis and biological evaluation of novel FGFR inhibitors bearing an indazole scaffold.
Org.Biomol.Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2015-05-13 |
| Resolution | 2.000 |
| CATH Insert Date | 28 Jun, 2015 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 29 Jun, 2015 | Chopped |
| B | 29 Jun, 2015 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4zsaA01 | 27 Jul, 2015 | 3.30.200.20 | Assigned |
| 4zsaA02 | 27 Jul, 2015 | 1.10.510.10 | Assigned |
| 4zsaB01 | 27 Jul, 2015 | 3.30.200.20 | Assigned |
| 4zsaB02 | 27 Jul, 2015 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P11362 | FGFR1_HUMAN | Homo sapiens | Fibroblast growth factor receptor 1 |
| P11362 | FGFR1_HUMAN | Homo sapiens | Fibroblast growth factor receptor 1 |
