PDB Information

PDB4ZG6
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Structural Basis for Inhibition of Human Autotaxin by Four Potent Compounds with Distinct Modes of Binding.
Stein, A.J., Bain, G., Prodanovich, P., Santini, A.M., Darlington, J., Stelzer, N.M., Sidhu, R.S., Schaub, J., Goulet, L., Lonergan, D., Calderon, I., Evans, J.F., Hutchinson, J.H.
Mol.Pharmacol.
HeaderHydrolase/Hydrolase Inhibitor
Released2015-04-22
Resolution1.800
CATH Insert Date25 Oct, 2015

PDB Images (11)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 26 Oct, 2015 Chopped
B 26 Oct, 2015 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
4zg6A01 31 Oct, 2015 Holding pen
4zg6A02 31 Oct, 2015 4.10.410.20 Assigned
4zg6A03 31 Oct, 2015 3.40.720.10 Assigned
4zg6A04 31 Oct, 2015 3.40.570.10 Assigned
4zg6B01 01 Nov, 2015 Holding pen
4zg6B02 01 Nov, 2015 4.10.410.20 Assigned
4zg6B03 01 Nov, 2015 3.40.720.10 Assigned
4zg6B04 01 Nov, 2015 3.40.570.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q13822 ENPP2_HUMAN Homo sapiens Ectonucleotide pyrophosphatase/phosphodiesterase family member 2
Q13822 ENPP2_HUMAN Homo sapiens Ectonucleotide pyrophosphatase/phosphodiesterase family member 2