PDB 4z22
PDB Information
| PDB | 4Z22 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Plasmodium falciparum |
| Primary Citation | Fragment-Based Discovery of 2-Aminoquinazolin-4(3H)-ones As Novel Class Nonpeptidomimetic Inhibitors of the Plasmepsins I, II, and IV.
J.Med.Chem.
|
| Header | Hydrolase |
| Released | 2015-03-28 |
| Resolution | 2.620 |
| CATH Insert Date | 10 Apr, 2016 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 11 Apr, 2016 | Chopped |
| B | 11 Apr, 2016 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4z22A01 | 02 May, 2016 | 2.40.70.10 | Assigned |
| 4z22A02 | 02 May, 2016 | 2.40.70.10 | Assigned |
| 4z22B01 | 02 May, 2016 | 2.40.70.10 | Assigned |
| 4z22B02 | 02 May, 2016 | 2.40.70.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P46925 | PLM2_PLAFA | Plasmodium falciparum | Plasmepsin-2 |
| P46925 | PLM2_PLAFA | Plasmodium falciparum | Plasmepsin-2 |
