PDB 4yyz
PDB Information
| PDB | 4YYZ |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli 'BL21-Gold(DE3)pLysS AG' |
| Gene Source | Homo sapiens |
| Primary Citation | Design of pyrozolo-pyrimidines as 11beta-HSD1 inhibitors through optimisation of molecular electrostatic potential.
Medchemcomm
|
| Header | Oxidoreductase |
| Released | 2015-03-24 |
| Resolution | 3.200 |
| CATH Insert Date | 10 Apr, 2016 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 11 Apr, 2016 | Chopped |
| B | 11 Apr, 2016 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4yyzA00 | 02 May, 2016 | 3.40.50.720 | Assigned |
| 4yyzB00 | 02 May, 2016 | 3.40.50.720 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P28845 | DHI1_HUMAN | Homo sapiens | Corticosteroid 11-beta-dehydrogenase isozyme 1 |
| P28845 | DHI1_HUMAN | Homo sapiens | Corticosteroid 11-beta-dehydrogenase isozyme 1 |
