PDB Information

PDB4Y5H
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Pyridopyrimidinone Derivatives as Potent and Selective c-Jun N-Terminal Kinase (JNK) Inhibitors.
Zheng, K., Park, C.M., Iqbal, S., Hernandez, P., Park, H., LoGrasso, P.V., Feng, Y.
Acs Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2015-02-11
Resolution2.060
CATH Insert Date28 Jun, 2015

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4y5hA01 22 Jul, 2015 3.30.200.20 Assigned
4y5hA02 22 Jul, 2015 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P53779 MK10_HUMAN Homo sapiens Mitogen-activated protein kinase 10