PDB Information

PDB4Y2H
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Aryl Pyrazoles as Potent Inhibitors of Arginine Methyltransferases: Identification of the First PRMT6 Tool Compound.
Mitchell, L.H., Drew, A.E., Ribich, S.A., Rioux, N., Swinger, K.K., Jacques, S.L., Lingaraj, T., Boriack-Sjodin, P.A., Waters, N.J., Wigle, T.J., Moradei, O., Jin, L., Riera, T., Porter-Scott, M., Moyer, M.P., Smith, J.J., Chesworth, R., Copeland, R.A.
Acs Med.Chem.Lett.
HeaderTransferase
Released2015-02-09
Resolution2.370
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4y2hA01 20 Jul, 2015 3.40.50.150 Assigned
4y2hA02 20 Jul, 2015 2.70.160.11 Assigned
4y2hB01 20 Mar, 2016 3.40.50.150 Assigned
4y2hB02 20 Mar, 2016 2.70.160.11 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q96LA8 ANM6_HUMAN Homo sapiens Protein arginine N-methyltransferase 6
Q96LA8 ANM6_HUMAN Homo sapiens Protein arginine N-methyltransferase 6