PDB 4y2b
PDB Information
| PDB | 4Y2B |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21(DE3) |
| Gene Source | Homo sapiens |
| Primary Citation | 2-(Isopropylamino)thieno[3,2-d]pyrimidin-4(3H)-one derivatives as selective phosphodiesterase 7 inhibitors with potent in vivo efficacy
Bioorg.Med.Chem.Lett.
|
| Header | Hydrolase/Hydrolase Inhibitor |
| Released | 2015-02-09 |
| Resolution | 2.200 |
| CATH Insert Date | 28 Jun, 2015 |
PDB Images (3)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 29 Jun, 2015 | Chopped |
CATH Domains (1)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4y2bA00 | 20 Jul, 2015 | 1.10.1300.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q13946 | PDE7A_HUMAN | Homo sapiens | High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A |
