PDB Information

PDB4XYF
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Discovery of Potent and Selective 8-Fluorotriazolopyridine c-Met Inhibitors.
Peterson, E.A., Teffera, Y., Albrecht, B.K., Bauer, D., Bellon, S.F., Boezio, A., Boezio, C., Broome, M.A., Choquette, D., Copeland, K.W., Dussault, I., Lewis, R., Lin, M.H., Lohman, J., Liu, J., Potashman, M., Rex, K., Shimanovich, R., Whittington, D.A., Vaida, K.R., Harmange, J.C.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2015-02-02
Resolution1.850
CATH Insert Date28 Jun, 2015

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4xyfA01 22 Jul, 2015 3.30.200.20 Assigned
4xyfA02 22 Jul, 2015 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P08581 MET_HUMAN Homo sapiens Hepatocyte growth factor receptor