PDB Information

PDB4XUZ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceKlebsiella pneumoniae subsp. pneumoniae
Primary Citation
Discovery of a Cyclic Boronic Acid beta-Lactamase Inhibitor (RPX7009) with Utility vs Class A Serine Carbapenemases.
Hecker, S.J., Reddy, K.R., Totrov, M., Hirst, G.C., Lomovskaya, O., Griffith, D.C., King, P., Tsivkovski, R., Sun, D., Sabet, M., Tarazi, Z., Clifton, M.C., Atkins, K., Raymond, A., Potts, K.T., Abendroth, J., Boyer, S.H., Loutit, J.S., Morgan, E.E., Durso, S., Dudley, M.N.
J.Med.Chem.
HeaderHydrolase/Antibiotic
Released2015-01-26
Resolution1.500
CATH Insert Date28 Jun, 2015

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4xuzA00 20 Jul, 2015 3.40.710.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
S5LVN3 S5LVN3_KLEPN Klebsiella pneumoniae subsp. pneumoniae Beta-lactamase