PDB Information

PDB4XUI
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceTrypanosoma cruzi
Primary Citation
Synthesis and Evaluation of Oxyguanidine Analogues of the Cysteine Protease Inhibitor WRR-483 against Cruzain.
Jones, B.D., Tochowicz, A., Tang, Y., Cameron, M.D., McCall, L.I., Hirata, K., Siqueira-Neto, J.L., Reed, S.L., McKerrow, J.H., Roush, W.R.
Acs Med.Chem.Lett.
HeaderHydrolase/Hydrolase Inhibitor
Released2015-01-26
Resolution2.510
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped
C 29 Jun, 2015 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
4xuiA00 20 Mar, 2016 3.90.70.10 Assigned
4xuiB00 20 Mar, 2016 3.90.70.10 Assigned
4xuiC00 20 Mar, 2016 3.90.70.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain