PDB 4xs3
PDB Information
| PDB | 4XS3 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Inhibition of Cancer-Associated Mutant Isocitrate Dehydrogenases by 2-Thiohydantoin Compounds.
J.Med.Chem.
|
| Header | Oxidoreductase/Oxidoreductase Inhibitor |
| Released | 2015-01-21 |
| Resolution | 3.290 |
| CATH Insert Date | 14 Aug, 2016 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 15 Aug, 2016 | Chopped |
| B | 15 Aug, 2016 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4xs3A00 | 01 Sep, 2016 | 3.40.718.10 | Assigned |
| 4xs3B00 | 01 Sep, 2016 | 3.40.718.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O75874 | IDHC_HUMAN | Homo sapiens | Isocitrate dehydrogenase [NADP] cytoplasmic |
| O75874 | IDHC_HUMAN | Homo sapiens | Isocitrate dehydrogenase [NADP] cytoplasmic |
