PDB Information

PDB4XJP
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMycobacterium tuberculosis (strain ATCC 25618 / H37Rv)
Primary Citation
Structure-Based Optimization of Pyridoxal 5'-Phosphate-Dependent Transaminase Enzyme (BioA) Inhibitors that Target Biotin Biosynthesis in Mycobacterium tuberculosis.
Liu, F., Dawadi, S., Maize, K.M., Dai, R., Park, S.W., Schnappinger, D., Finzel, B.C., Aldrich, C.C.
J. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2015-01-08
Resolution1.600
CATH Insert Date10 Apr, 2016

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Chopped
B 11 Apr, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4xjpA01 29 Apr, 2016 3.90.1150.10 Assigned
4xjpA02 29 Apr, 2016 3.40.640.10 Assigned
4xjpB01 29 Apr, 2016 3.90.1150.10 Assigned
4xjpB02 29 Apr, 2016 3.40.640.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P9WQ81 BIOA_MYCTU Mycobacterium tuberculosis H37Rv Adenosylmethionine-8-amino-7-oxononanoate aminotransferase
P9WQ81 BIOA_MYCTU Mycobacterium tuberculosis H37Rv Adenosylmethionine-8-amino-7-oxononanoate aminotransferase