PDB Information

PDB4X7Q
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-based design of low-nanomolar PIM kinase inhibitors.
Ishchenko, A., Zhang, L., Le Brazidec, J.Y., Fan, J., Chong, J.H., Hingway, A., Raditsis, A., Singh, L., Elenbaas, B., Hong, V.S., Marcotte, D., Silvian, L., Enyedy, I., Chao, J.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2014-12-09
Resolution2.330
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4x7qA01 22 Jul, 2015 3.30.200.20 Assigned
4x7qA02 22 Jul, 2015 1.10.510.10 Assigned
4x7qB01 22 Jul, 2015 3.30.200.20 Assigned
4x7qB02 22 Jul, 2015 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9P1W9 PIM2_HUMAN Homo sapiens Serine/threonine-protein kinase pim-2
Q9P1W9 PIM2_HUMAN Homo sapiens Serine/threonine-protein kinase pim-2