PDB 4x2u
PDB Information
| PDB | 4X2U |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Plasmodium falciparum FcB1/Columbia |
| Primary Citation | X-ray crystal structures of an orally available aminopeptidase inhibitor, Tosedostat, bound to anti-malarial drug targets PfA-M1 and PfA-M17.
Proteins
|
| Header | Hydrolase/Hydrolase Inhibitor |
| Released | 2014-11-27 |
| Resolution | 1.500 |
| CATH Insert Date | 28 Jun, 2015 |
PDB Images (7)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 29 Jun, 2015 | Chopped |
CATH Domains (5)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4x2uA01 | 20 Jul, 2015 | 2.60.40.1730 | Assigned |
| 4x2uA02 | 20 Jul, 2015 | 3.30.2010.30 | Assigned |
| 4x2uA03 | 20 Jul, 2015 | 1.10.390.10 | Assigned |
| 4x2uA04 | 20 Jul, 2015 | 2.60.40.1840 | Assigned |
| 4x2uA05 | 20 Jul, 2015 | 1.25.50.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O96935 | AMP1_PLAFQ | Plasmodium falciparum FcB1/Columbia | M1 family aminopeptidase |
