PDB Information

PDB4WHL
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
A new class of peptidomimetics targeting the polo-box domain of polo-like kinase 1.
Ahn, M., Han, Y.H., Park, J.E., Kim, S., Lee, W.C., Lee, S.J., Gunasekaran, P., Cheong, C., Shin, S.Y., Kim, H.Y., Ryu, E.K., Murugan, R.N., Kim, N.H., Bang, J.K.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2014-09-23
Resolution2.710
CATH Insert Date21 Dec, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 22 Dec, 2014 Chopped
B 22 Dec, 2014 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4whlA01 29 Dec, 2014 3.30.1120.30 Assigned
4whlA02 29 Dec, 2014 3.30.1120.30 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P53350 PLK1_HUMAN Homo sapiens Serine/threonine-protein kinase PLK1